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6. Tutorial Sheet 1

The document consists of tutorial sheets for the subject Medicinal Chemistry III and PH Biotechnology, covering various topics such as beta-lactam antibiotics, anti-tubercular drugs, urinary tract anti-infective agents, antifungal antibiotics, and drug design. Each sheet contains questions related to classification, mechanism of action, synthesis, structure, and uses of different pharmaceutical compounds. The tutorials are designed for pharmacy students to enhance their understanding and knowledge in medicinal chemistry.

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Vinay ghalout
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15 views

6. Tutorial Sheet 1

The document consists of tutorial sheets for the subject Medicinal Chemistry III and PH Biotechnology, covering various topics such as beta-lactam antibiotics, anti-tubercular drugs, urinary tract anti-infective agents, antifungal antibiotics, and drug design. Each sheet contains questions related to classification, mechanism of action, synthesis, structure, and uses of different pharmaceutical compounds. The tutorials are designed for pharmacy students to enhance their understanding and knowledge in medicinal chemistry.

Uploaded by

Vinay ghalout
Copyright
© © All Rights Reserved
We take content rights seriously. If you suspect this is your content, claim it here.
Available Formats
Download as PDF, TXT or read online on Scribd
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BUDDHA INSTITUTE OF PHARMCY

GIDA, GORAKHPUR
TUTORIAL SHEET-1
SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar
SUB. CODE: BP 601T UNIT: 1
BRANCH: PHARMACY. TOPIC: Beta lactam antibiotics

Q.1: Write down the classification, mechanism of action and


structural activity relationship of the following drugs(AKTU 2018)
a) Penicillin
b) Cephalosporin
Q.2 Write down the classification, mechanism of action and
structural activity relationship of the following drugs(AKTU2017)
A) Monobactam
B) Streptomycin
C) Neomycin
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-2
SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar
SUB. CODE: BP 601T UNIT: 1
BRANCH: PHARMACY. TOPIC: Beta lactam antibiotics

Q.1: Write a note on beta lactam inhibitors and


monobactam.(AKTU2022)
Q.2: Give the classification, mechanism of action and uses of
aminoglycosides antibiotics.(AKTU2022)

Q.3 Give the classification tetracyclin SAR and use of it(AKTU


2022)
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-3

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 2
BRANCH: PHARMACY. TOPIC:Macrolides

Q.1: Write down the synthesis, structure, mechanism of action


and SAR of chloramphenicol. (AKTU 2023)
Q.2: Write a short note on prodrug.(AKTU2023)
Q.3. Give the structure of Azithromycin, clarithromycin,
kanamycin. (AKTU2019)
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-4

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 2
BRANCH: PHARMACY. TOPIC: Malarial
Drug

Q.1: Write a short note on malaria.(AKTU2022)


Q.2: Give the synthesis, mechanism of action, SAR and uses of
chloroquine.(AKTU2022)
Q.3. Write down the structure of the following(AKTU2018)
a) Pamaquine b) Mefloquine
c) Cycloguanil pamoate d) Atovoquone
Q.4. Define and classify bigunides with example and use of it.
Q.5 Give the structure of pyrimethamine, atovaquone.(AKTU
2022)
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-5
SUBJECT: PH BIOTECHNOLOGY NAME OF FACULTY: Vinay Kumar
SUB. CODE: BP 601T UNIT: 3
BRANCH: PHARMACY. TOPIC: Anti tubercular drug

Q.1: Define and classify anti tubercular agent.(AKTU2018)


Q.2.Give the synthesis and use of isoniazid and para amino
salicylic acid.(AKTU2019)
Q.3. Give the structure of the following-(AKTU2017)
a) Ethionamide b) Cycloserine c) streptomycin d) Pyrazinamide
Q.4. Write a short note on anti tuberculae agent.(2019)
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-6

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 3
BRANCH: PHARMACY TOPIC: Urinary tract anti infective agent

Q.1: Give the classification of urinary tract anti-infective agent


with example.(AKTU2021)
Q.2: Write down the SAR of quinolones.(AKTU2022)
Q.3. Give the synthesis of the following-(AKTU2017)
a) Ciprofloxacin b) Acyclovir
Q.4. Give the classification of antiviral agent.(AKTU2022)
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-7

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 4
BRANCH: PHARMACY TOPIC: Antifungal Antibiotics

Q.1: Give the classification of antifungal antibiotics with


example.(AKTU2018)
Q.2: Write down the structure of the following-(AKTU2019)

a) Clotrimazole
b) Econazole
c) Ketoconazole
d) Intraconazole
Q.3. Give the synthesis, MOA and uses of the following-
(AKTU2022)
a) Metronidazole b) Mebendazole
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-8

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 4
BRANCH: PHARMACY TOPIC: Antifungal Antibiotics

Q.1: Give the classification of anti protozoal agent with


example.(AKTU2016)
Q.2: Give the SAR of sulphones and synthesis of
sulphamethaxazole.(AKTU2023)
Q. 3. Give the structure of clotrimazole, econazole,
ketoconazole.(AKTU 2021)
Q.4. Give the structure of the following-(AKTU 2019)
A) Intraconazole C) Fluconazole
B) Tinidazole D)Albendazole
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-9

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 5
BRANCH: PHARMACY TOPIC: Drug Design

Q.1: Write a short note on introduction of drug


design.(AKTU2023)
Q.2: What is the physiological parameter of used in
QSAR?(AKTU2018)
Q.3: What is the application of drug designing?(AKTU2022)
BUDDHA INSTITUTE OF PHARMCY
GIDA, GORAKHPUR
TUTORIAL SHEET-10

SUBJECT: Medicinal Chemistry III NAME OF FACULTY: Vinay Kumar


SUB. CODE: BP 601T UNIT: 5
BRANCH: PHARMACY TOPIC: Drug Design

Q.1: What is pharmacophore modeling and explain in short


about docking technique?(AKTU2021)
Q.2: Give the application of combinatorial
chemistry.(AKTU2021)
Q.3. Define combinatorial chemistry and what are the
significance of it?(AKTU2022)

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